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Found 3 Enz. Inhib. hit(s) with Target = 'Hydroxycarboxylic acid receptor 2' and Ligand = 'BDBM50208122'
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50208122((+)-5-(5-chloro-thiophen-3-yl)-5-methyl-4-oxo-4,5-...)
Affinity DataEC50:  4.68E+3nMAssay Description:Activity at GPR109a in CHO cells assessed as inhibition of forskolin-induced cAMP generationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50208122((+)-5-(5-chloro-thiophen-3-yl)-5-methyl-4-oxo-4,5-...)
Affinity DataEC50:  200nMAssay Description:Activity at GPR109a (unknown origin) assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50208122((+)-5-(5-chloro-thiophen-3-yl)-5-methyl-4-oxo-4,5-...)
Affinity DataEC50:  4.68E+3nMAssay Description:Activity at GPR109a in CHO cells assessed as inhibition of forskolin-induced cAMP generationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed