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Found 3 Enz. Inhib. hit(s) with Target = 'Integrase' and Ligand = 'BDBM50409847'
TargetIntegrase(Human immunodeficiency virus 1)TBA
LigandPNGBDBM50409847(CHEMBL131784)
Affinity DataIC50:  4.26E+3nMAssay Description:Inhibition of Human immunodeficiency virus 1 integrase strand transfer activity using [32P]5'end-labeled linear 21 mer as substrate incubated for 30 ...More data for this Ligand-Target Pair
In DepthDetails Article
TargetIntegrase(Human immunodeficiency virus 1)
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50409847(CHEMBL131784)
Affinity DataIC50:  7.41E+3nMAssay Description:Inhibitory activity against DNA strand transfer by HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
University Of Southern California

Curated by ChEMBL
LigandPNGBDBM50409847(CHEMBL131784)
Affinity DataIC50:  9.33E+3nMAssay Description:Inhibitory activity against 3' processing by HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed