BindingDB PrimarySearch

Found 1 Enz. Inhib. hit(s) with Target = 'Isoform C of Bromodomain-containing protein 4 (Short)' and Ligand = 'BDBM50380682'

Isoform C of Bromodomain-containing protein 4 (Short)(Homo sapiens (Human))
Dana-Farber Cancer Institute

BDBM50380682(CHEMBL2017291 | I-BET151 (16))

IC50: 29.4nMpH: 7.5 T: 2°CAssay Description:Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150...More data for this Ligand-Target Pair

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3D Structure (crystal)