Affinity DataKi: 0.840nMAssay Description:Binding affinity against cloned human opioid Opioid receptor kappa 1 transfected onto CHO cells using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor kappa 1 (U-69,593) transfected onto CHO cellsMore data for this Ligand-Target Pair