Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50157799'
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50157799(1'-benzyl-6,7-didehydro-3,14-dihydroxy-4,5alpha-ep...)
Affinity DataKi:  289nMAssay Description:Displacement of [3H]U-69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bath

Curated by ChEMBL
LigandPNGBDBM50157799(1'-benzyl-6,7-didehydro-3,14-dihydroxy-4,5alpha-ep...)
Affinity DataEC50:  1.75E+3nMAssay Description:Activity at human recombinant kappa opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed