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Found 4 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50297347'
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50297347((2S,5S,8S,13S,Z)-13-((S)-2-(2-(2-((S)-2-amino-3-(4...)
Affinity DataKi:  2.46nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50297347((2S,5S,8S,13S,Z)-13-((S)-2-(2-(2-((S)-2-amino-3-(4...)
Affinity DataKi:  10.9nMAssay Description:Displacement of [3H]Diprenorphine from rat kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50297347((2S,5S,8S,13S,Z)-13-((S)-2-(2-(2-((S)-2-amino-3-(4...)
Affinity DataEC50:  8.30nMAssay Description:Agonist activity at rat cloned kappa opioid receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50297347((2S,5S,8S,13S,Z)-13-((S)-2-(2-(2-((S)-2-amino-3-(4...)
Affinity DataEC50:  23nMAssay Description:Agonist activity at rat cloned kappa opioid receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP production by scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed