Affinity DataKi: 4.40nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cells by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 136nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO cells assessed as [35S]GTPgammaS binding by scintillation counting analysisMore data for this Ligand-Target Pair