Affinity DataKi: 153nMAssay Description:Compound was evaluated for the inhibition of [3H]-bremazocine binding to Opioid receptor kappa 1 in guinea pig cerebellum membrane homogenates.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was evaluated for the agonistic activity against Opioid receptor kappa 1 in rabbit vas deferens.More data for this Ligand-Target Pair