Report error Found 3 Enz. Inhib. hit(s) with Target = 'KiSS-1 receptor' and Ligand = 'BDBM50045514'
Affinity DataKi: 0.0260nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Agonist activity at rat KISS1R transfected in CHO cells assessed as intracellular calcium flux after 24 hrs by functional FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.440nMAssay Description:Agonist activity at human KISS1R transfected in CHO cells assessed as intracellular calcium flux after 24 hrs by functional FLIPR assayMore data for this Ligand-Target Pair