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Found 3 Enz. Inhib. hit(s) with Target = 'Kinesin-like protein KIF11' and Ligand = 'BDBM50382582'
TargetKinesin-like protein KIF11(Homo sapiens (Human))
The Beatson Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50382582(CHEMBL2022999)
Affinity DataKi:  7.5nMAssay Description:Inhibition of N-terminal hexa-histidine tagged human cloned Eg5 (1 to 368 amino acids) expressed in Escherichia coli BL21 (DE3) assessed as reduction...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
The Beatson Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50382582(CHEMBL2022999)
Affinity DataKi:  9.80nMAssay Description:Inhibition of N-terminal hexa-histidine tagged human cloned Eg5 (1 to 368 amino acids) expressed in Escherichia coli BL21 (DE3) assessed as reduction...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
The Beatson Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50382582(CHEMBL2022999)
Affinity DataEC50:  95nMAssay Description:Inhibition of N-terminal hexa-histidine tagged human cloned Eg5 (1 to 368 amino acids) expressed in Escherichia coli BL21 (DE3) assessed as reduction...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed