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Found 4 Enz. Inhib. hit(s) with Target = 'Leucine-rich repeat serine/threonine-protein kinase 2' and Ligand = 'BDBM50603018'
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50603018(CHEMBL5200822)
Affinity DataIC50:  5nMAssay Description:Inhibition of full length LRRK2 G2019S mutant (unknown origin) by LRRKtide Adapta assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50603018(CHEMBL5200822)
Affinity DataIC50:  22nMAssay Description:Inhibition of full length wild type LRRK2 (unknown origin) by LRRKtide Adapta assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50603018(CHEMBL5200822)
Affinity DataEC50:  620nMAssay Description:Inhibition of pcDNA5FRT-TO-GFP fused - LRRK2 G2019S mutant (unknown origin) transfected in HEK293 cells incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Stanford University

Curated by ChEMBL
LigandPNGBDBM50603018(CHEMBL5200822)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of wild type pcDNA5FRT-TO-GFP fused - LRRK2 (unknown origin) transfected in HEK293 cells incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed