Found 6 Enz. Inhib. hit(s) with Target = 'Lysophosphatidic acid receptor 1' and Ligand = 'BDBM50148348'
Affinity DataEC50: 17nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: 350nMAssay Description:Agonist activity at human LPA1 expressed in LPA1xLPA2 double knockout mouse MEF cells up to 10 uM by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
Affinity DataKd: 5.60nMAssay Description:Binding affinity to LPA1 receptor (unknown origin) by cell-based backscattering interferometryMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 830nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
Affinity DataEC50: 31nMAssay Description:Agonist activity at LPA1 expressed in human chem1 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair