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Found 2 Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50189576'
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50189576((R)-6-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3...)
Affinity DataKi:  3.30nMAssay Description:Binding affinity to chimeric rat/human MCH1R stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50189576((R)-6-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3...)
Affinity DataIC50:  7.70nMAssay Description:Activity at chimeric rat/human MCH1R by accumulation of GTPgammaSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed