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Found 2 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 3' and Ligand = 'BDBM50184363'
TargetMelanocortin receptor 3(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184363(CHEMBL263822 | c[Nle-Arg-D-Phe-Arg-Trp-Glu]-NH2)
Affinity DataIC50:  140nMAssay Description:Inhibitory activity against hMC3R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184363(CHEMBL263822 | c[Nle-Arg-D-Phe-Arg-Trp-Glu]-NH2)
Affinity DataEC50:  1.20nMAssay Description:Activity against hMC3R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed