Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50033134'
TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50033134((3R,6S,9R,12S,15S,23R)-15-((S)-2-Acetylamino-hexan...)
Affinity DataKi:  20nMAssay Description:Binding affinity against human melanocortin receptor 4 (hMC4R) (concentration of the peptide at 50% specific binding)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50033134((3R,6S,9R,12S,15S,23R)-15-((S)-2-Acetylamino-hexan...)
Affinity DataIC50:  1.80nMAssay Description:Inhibitory activity against human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50033134((3R,6S,9R,12S,15S,23R)-15-((S)-2-Acetylamino-hexan...)
Affinity DataKd:  0.501nMAssay Description:Evaluated for agonist activity at cloned mammalian Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed