Affinity DataKi: 860nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-5 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 326nMAssay Description:Concentration required for 50% inhibition by displacement of of [125I]NDP-alpha-MSH of human MC5R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 326nMAssay Description:Evaluated for binding affinity against human melanocortin 5 (hMC5R) receptor by displacing [125I]-NDP-alpha-MSH radioligand expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 326nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC5R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+3nMAssay Description:Evaluated for binding affinity against rat Melanocortin-5 receptor (rMC5R) by displacing [125I]NDP-alpha-MSH radioligand expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 737nMAssay Description:Functional activity as concentration at 50% maximum cAMP accumulation in human melanocortin 1 (MC5R) receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 736nMAssay Description:Evaluated for Functional Activity at MC5R as effective concentration at 50% maximum CMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+3nMAssay Description:Functional activity as concentration of the compound at 50% maximum cAMP accumulation in rat Melanocortin-5 receptor (rMC5R)More data for this Ligand-Target Pair
Affinity DataEC50: 737nMAssay Description:Activity against human MC5R by cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+3nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair