Found 15 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 5' and Ligand = 'BDBM50184359' 
Affinity DataIC50: 4.20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by Wallac 1470 gamma countingMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:Displacement of [125I][Nle4,Dphe7]-alpha-MSH from human MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibitory concentration against human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
Affinity DataEC50: 0.160nMAssay Description:Agonist activity towards mouse Melanocortin-5 receptor (mMC5R)More data for this Ligand-Target Pair
Affinity DataEC50: 0.160nMAssay Description:Activity in mouse melanocortin-5 receptor stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 5.70nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 8nMAssay Description:Activity at human MC5R expressed in HEK293 cells assessed by measuring intracellular cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:Activity against hMC5R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Effective concentration that was able to generate 50% maximal intracellular cAMP in L-cells transfected with Melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Agonistic activity against human melanocortin receptor (hMC5R) for cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as stimulation of intracellular cAMP levelMore data for this Ligand-Target Pair
