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Found 2 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 5' and Ligand = 'BDBM50184360'
TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184360(CHEMBL204864 | c[Nle-Nle-D-Nal(2')-Arg-Trp-Glu]-NH...)
Affinity DataIC50:  3.80nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184360(CHEMBL204864 | c[Nle-Nle-D-Nal(2')-Arg-Trp-Glu]-NH...)
Affinity DataEC50:  200nMAssay Description:Activity against hMC5R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed