TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Naples "Federico Ii
Curated by ChEMBL
University Of Naples "Federico Ii
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair