Found 3 Enz. Inhib. hit(s) with Target = 'Melatonin receptor type 1A/1B' and Ligand = 'BDBM50230659'
Affinity DataKi: 2.20nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to melatonin receptor in quail brain as 1/KaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0000500nMAssay Description:Monophasic inhibitory concentration against melatonin receptor was measured on ovine pars tuberalis membrane.More data for this Ligand-Target Pair
Affinity DataKd: 0.000453nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair