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Found 4 Enz. Inhib. hit(s) with Target = 'Melatonin receptor type 1A/1B' and Ligand = 'BDBM50471112'
TargetMelatonin receptor type 1A/1B(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50471112(CHEMBL61991)
Affinity DataKi:  0.390nMAssay Description:Binding affinity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin as labelled ligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50471112(CHEMBL61991)
Affinity DataIC50:  1.10nMAssay Description:Inhibitory activity against melatonin receptor of quail optica tecta with 200 pM 2-[125] iodomelatoninMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50471112(CHEMBL61991)
Affinity DataIC50:  1.40nMAssay Description:Inhibitory activity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin as radiolabeled ligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50471112(CHEMBL61991)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against melatonin receptor of quail optica tecta with 200 pM 2-[125] iodomelatonin as gamma-S (10e-4 M)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed