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Found 3 Enz. Inhib. hit(s) with Target = 'Melatonin receptor type 1B' and Ligand = 'BDBM50155730'
TargetMelatonin receptor type 1B(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50155730(1-[1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydr...)
Affinity DataKi:  9.80nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to human melatonin receptor MT2 expressed in NIH3T3 rat fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50155730(1-[1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydr...)
Affinity DataIC50:  9.70nMAssay Description:Antagonist activity at MT2 receptor (unknown origin) assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50155730(1-[1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydr...)
Affinity DataIC50:  9.70nMAssay Description:Inhibitory concentration against Melatonin receptor type 1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed