Affinity DataKi: 9.80nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to human melatonin receptor MT2 expressed in NIH3T3 rat fibroblast cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.70nMAssay Description:Antagonist activity at MT2 receptor (unknown origin) assessed as cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 9.70nMAssay Description:Inhibitory concentration against Melatonin receptor type 1BMore data for this Ligand-Target Pair