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Found 1 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 14' and Ligand = 'BDBM552793'
TargetMitogen-activated protein kinase kinase kinase 14(Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM552793((R)-7-(3-(2-(7H-Pyrrolo[2,3-b]pyrimidin-5-yl)thiaz...)
Affinity DataIC50: <100nMAssay Description:NIK/MAP3K14 auto-phosphorylation activity was measured using the AlphaScreenŽ (ascreen) format (Perkin Elmer). All compound6 tested were dissolved in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed