Found 6 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50000518' TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute of Montreal
Curated by ChEMBL
Clinical Research Institute of Montreal
Curated by ChEMBL
Affinity DataKi: 143nMAssay Description:Inhibition of [3H]- ]DAMGO binding to mu receptor from rat brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute of Montreal
Curated by ChEMBL
Clinical Research Institute of Montreal
Curated by ChEMBL
Affinity DataKi: 336nMAssay Description:Binding affinity against Opioid receptor mu 1 in P2 membrane preparation of rat brain by [3H]DAGO displacement.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute of Montreal
Curated by ChEMBL
Clinical Research Institute of Montreal
Curated by ChEMBL
Affinity DataKi: 344nMAssay Description:Compound was tested for its binding affinity against opioid receptor mu using [3H]-DAGO as radioligand.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute of Montreal
Curated by ChEMBL
Clinical Research Institute of Montreal
Curated by ChEMBL
Affinity DataKi: 415nMAssay Description:Inhibition of [3H]- ]DAMGO binding to mu receptor from rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 281nMAssay Description:Inhibition of electrically evoked contractions in Guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 4.42E+3nMAssay Description:Inhibition of electrically evoked contractions in Guinea pig ileumMore data for this Ligand-Target Pair
