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Found 5 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50068132'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50068132(3-[(4-Benzyl-piperazin-1-yl)-(4-tert-butyl-phenyl)...)
Affinity DataIC50:  1.10E+4nMAssay Description:Binding affinity was measured against Opioid receptor mu 1 using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50068132(3-[(4-Benzyl-piperazin-1-yl)-(4-tert-butyl-phenyl)...)
Affinity DataIC50:  1.10E+4nMAssay Description:Binding affinity was measured against Opioid receptor mu 1 using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50068132(3-[(4-Benzyl-piperazin-1-yl)-(4-tert-butyl-phenyl)...)
Affinity DataIC50:  1.70E+4nMAssay Description:In vitro inhibition of [3H]-DAMGO (Tyr-D-Ala-Gly-(Me)-Phe-Gly-ol) binding to Opioid receptor mu 1 using rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50068132(3-[(4-Benzyl-piperazin-1-yl)-(4-tert-butyl-phenyl)...)
Affinity DataEC50:  7.60E+3nMAssay Description:Tested for electrically induced smooth muscle contractions from guinea pig ileum expressed in mu opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
The University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50068132(3-[(4-Benzyl-piperazin-1-yl)-(4-tert-butyl-phenyl)...)
Affinity DataEC50:  3.90E+4nMAssay Description:Tested for electrically induced smooth muscle contractions from guinea pig ileum expressed in mu opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed