Affinity DataKi: 2.20nMAssay Description:Inhibition of stimulation of [35S]GTP-gamma-S, binding produced by the selective agonist (DAMGO, mu-receptor), in guinea pig caudate membranes.More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Antagonist activity on agonist (DAMGO) stimulated [35S]GTP-gamma-S, binding in cloned mu opioid receptors.More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity to mu-opioid receptor of rat brain using [3H]DAMGO as radioligand.More data for this Ligand-Target Pair