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Found 2 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50257774'
TargetMu-type opioid receptor(Homo sapiens (Human))
Alkem Laboratories

Curated by ChEMBL
LigandPNGBDBM50257774(CHEMBL4104814)
Affinity DataIC50:  780nMAssay Description:Antagonist activity at recombinant human MOR expressed in HEK293T cells assessed as reduction in DAMGO-induced inhibition of forskolin-stimulated cAM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Alkem Laboratories

Curated by ChEMBL
LigandPNGBDBM50257774(CHEMBL4104814)
Affinity DataIC50:  794nMAssay Description:Antagonist activity at recombinant human MOR expressed in HEK293T cells assessed as reduction in DAMGO-induced inhibition of forskolin-stimulated cAM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed