Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor' and Ligand = 'BDBM50004725'
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50004725(1,3-Dimethyl-1-(1-methyl-4-pyrrolidin-1-yl-but-2-y...)
Affinity DataKd:  7.50E+3nMAssay Description:Inhibition of Shh signaling in mouse Shh-light2 cells by Gli-dependent firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50004725(1,3-Dimethyl-1-(1-methyl-4-pyrrolidin-1-yl-but-2-y...)
Affinity DataEC50:  2.11E+3nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed