Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1/M2/M3/M4/M5' and Ligand = 'BDBM50004733'
LigandPNGBDBM50004733(1-Methyl-3-(4-pyrrolidin-1-yl-but-2-ynyl)-imidazol...)
Affinity DataKi:  2.70nMAssay Description:Binding affinity to muscarinic acetylcholine receptor was determined in presence of [3H]OXO-M radioligand (in vitro)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50004733(1-Methyl-3-(4-pyrrolidin-1-yl-but-2-ynyl)-imidazol...)
Affinity DataKi:  180nMAssay Description:Binding affinity to muscarinic acetylcholine receptor was determined in presence of [3H]QNB radioligand (in vitro)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50004733(1-Methyl-3-(4-pyrrolidin-1-yl-but-2-ynyl)-imidazol...)
Affinity DataKi:  1.60E+3nMAssay Description:Muscarinic acetylcholine receptor M3 agonistic/antagonistic activity in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed