Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50450592'
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]pirenzepine from muscarinic M1 receptor of rat cortex homogenates.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKi:  0.150nMAssay Description:Ability to displace [3H]pirenzepine (PZ) from M1 receptor in rat cortex homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]pirenzepine from muscarinic acetylcholine receptor M1 in rat cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKd:  0.320nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 using [3H]QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed