Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50038212'
TargetMuscarinic acetylcholine receptor M2(RAT)
Institute For Drug Discovery Research
Curated by ChEMBL
Institute For Drug Discovery Research
Curated by ChEMBL
Affinity DataKi: 970nMAssay Description:Compound tested in vitro for displacement of [3H]quinuclidinyl benzilate from rat cerebellum membrane expressing muscarinic M2 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:M2 agonist activity estimated by depression of isolated guinea pig left atriumMore data for this Ligand-Target Pair