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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50095103'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))TBA
LigandPNGBDBM50095103(4-{2-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenyl]-tet...)
Affinity DataKi:  5nMAssay Description:Antagonist activity at muscarinic M2 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))TBA
LigandPNGBDBM50095103(4-{2-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenyl]-tet...)
Affinity DataKi:  5.10nMAssay Description:Binding affinity at human cloned acetylcholine receptor M2 in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed