Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50208043'
Affinity DataKi: 21.9nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Activity at muscarinic M2 receptor in Albino Dunkin-Hartley guinea pig left atria assessed as inhibition of methacholine-induced bradycardiaMore data for this Ligand-Target Pair