Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M3' and Ligand = 'BDBM81900'
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM81900(AQ-RA 741 | CAS_129989 | NSC_129989)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]-NMS from human muscarinic M3 receptor expressed in stable CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM81900(AQ-RA 741 | CAS_129989 | NSC_129989)
Affinity DataKi:  63.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Regensburg

Curated by ChEMBL
LigandPNGBDBM81900(AQ-RA 741 | CAS_129989 | NSC_129989)
Affinity DataKi:  100nMAssay Description:Binding affinity to muscarinic M3 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
University of Bologna

Curated by PDSP Ki Database
LigandPNGBDBM81900(AQ-RA 741 | CAS_129989 | NSC_129989)
Affinity DataKi:  158nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed