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Found 8 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M4' and Ligand = 'BDBM50071173'
TargetMuscarinic acetylcholine receptor M4(bovine)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM50071173((3R,4R,4aS,8aR)-4-[(E)-2-((2S,6S)-1,6-Dimethyl-pip...)
Affinity DataKi:  2.95nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM50071173((3R,4R,4aS,8aR)-4-[(E)-2-((2S,6S)-1,6-Dimethyl-pip...)
Affinity DataKi:  6.02nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Chick)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM50071173((3R,4R,4aS,8aR)-4-[(E)-2-((2S,6S)-1,6-Dimethyl-pip...)
Affinity DataKi:  6.31nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
National Institute of Neurological Disorders and Stroke

Curated by PDSP Ki Database
LigandPNGBDBM50071173((3R,4R,4aS,8aR)-4-[(E)-2-((2S,6S)-1,6-Dimethyl-pip...)
Affinity DataKi:  11.0nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(bovine)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM50071173((3R,4R,4aS,8aR)-4-[(E)-2-((2S,6S)-1,6-Dimethyl-pip...)
Affinity DataKi:  11.7nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM50071173((3R,4R,4aS,8aR)-4-[(E)-2-((2S,6S)-1,6-Dimethyl-pip...)
Affinity DataKi:  46nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM50071173((3R,4R,4aS,8aR)-4-[(E)-2-((2S,6S)-1,6-Dimethyl-pip...)
Affinity DataKi:  50nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(MOUSE)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50071173((3R,4R,4aS,8aR)-4-[(E)-2-((2S,6S)-1,6-Dimethyl-pip...)
Affinity DataKi:  60nMMore data for this Ligand-Target Pair
In DepthDetails PubMed