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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M5' and Ligand = 'BDBM50231856'
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50231856(CHEMBL271519 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO-K1 cells assessed as inhibition of acetylcholine-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(RAT)
Vanderbilt Institute Of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50231856(CHEMBL271519 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M5 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed