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Found 2 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-3' and Ligand = 'BDBM50254482'
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Copenhagen University

Curated by ChEMBL
LigandPNGBDBM50254482(3-(dimethylamino)butyl benzyl(methyl)carbamate | C...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Copenhagen University

Curated by ChEMBL
LigandPNGBDBM50254482(3-(dimethylamino)butyl benzyl(methyl)carbamate | C...)
Affinity DataEC50:  6.70E+3nMAssay Description:Agonist activity at alpha3beta4 nAChR (unknown origin) expressed in HEK293 cells by FLIPR membrane potential assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed