Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4' and Ligand = 'BDBM50254538'
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Copenhagen University

Curated by ChEMBL
LigandPNGBDBM50254538(3-(dimethylamino)butyl methylcarbamate | CHEMBL466...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50254538(3-(dimethylamino)butyl methylcarbamate | CHEMBL466...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]epibatidine from rat recombinant alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50254538(3-(dimethylamino)butyl methylcarbamate | CHEMBL466...)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [3H]epibatidine from rat recombinant alpha-4-beta-4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed