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Found 2 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4' and Ligand = 'BDBM50254541'
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Copenhagen University

Curated by ChEMBL
LigandPNGBDBM50254541(5-(dimethylamino)-N,N-dimethylhex-2-enamide | CHEM...)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Copenhagen University

Curated by ChEMBL
LigandPNGBDBM50254541(5-(dimethylamino)-N,N-dimethylhex-2-enamide | CHEM...)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]epibatidine from alpha4beta4 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed