Found 2 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-7' and Ligand = 'BDBM50016185'
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Critical Therapeutics
Curated by ChEMBL
Critical Therapeutics
Curated by ChEMBL
Affinity DataEC50: 200nMAssay Description:Agonist activity at human alpha7 nAChR expressed in Xenopus oocytes by voltage clamp methodMore data for this Ligand-Target Pair