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Found 3 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-7' and Ligand = 'BDBM50082081'
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50082081(CHEMBL3422581)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR transfected in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50082081(CHEMBL3422581)
Affinity DataEC50:  145nMAssay Description:Agonist activity at rat alpha7 nAChR expressed in GH4C1 cells by fluorescent calcium assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50082081(CHEMBL3422581)
Affinity DataEC50:  2.73E+4nMAssay Description:Agonist activity at rat alpha7 nAChR expressed in GH4C1 cells by patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed