Found 1 Enz. Inhib. hit(s) with Target = 'Nuclear factor erythroid 2-related factor 2' and Ligand = 'BDBM50535743'
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Dongguk University
Curated by ChEMBL
Dongguk University
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of NRF2 in human MDA-MB-231 cells harboring ARE-GFP-Luc assessed as reduction in ARE-luciferase activity after 16 hrs by firefly luciferas...More data for this Ligand-Target Pair