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Found 4 Enz. Inhib. hit(s) with Target = 'Nuclear receptor ROR-gamma' and Ligand = 'BDBM50108881'
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50108881(CHEMBL3596591)
Affinity DataIC50:  220nMAssay Description:Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50108881(CHEMBL3596591)
Affinity DataIC50:  220nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50108881(CHEMBL3596591)
Affinity DataEC50:  200nMAssay Description:Inverse agonist activity at human ROR-gamma transfected in HEK293T cells by Gal4 luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50108881(CHEMBL3596591)
Affinity DataEC50:  200nMAssay Description:Inverse agonist activity at Gal4 DNA binding domain-tagged human RORgammat expressed in HEK293T cells assessed as effect on receptor-mediated transcr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed