Found 5 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 1 group D member 1' and Ligand = 'BDBM50383684' TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataEC50: 500nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataEC50: 2.30E+3nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataEC50: 2.30E+3nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataEC50: 2.30E+3nMAssay Description:Agonist activity at Rev-Erbalpha expressed in HEK293 cells coexpressing BamII promoter assessed as repression of transcription after 24 hrs by dual-G...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataEC50: 400nMAssay Description:Agonist activity at Rev-erbalpha assessed as NCoR recruitment by FRET assayMore data for this Ligand-Target Pair
