Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 1 group I member 2' and Ligand = 'BDBM50527154'
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50527154(CHEMBL4454255)
Affinity DataEC50:  5.70E+3nMAssay Description:Transactivation of human PXR transfected in human HepG2 cells co-transfected with CYP3A4-Luc plasmid incubated for overnight by luciferase reporter g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB