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Found 3 Enz. Inhib. hit(s) with Target = 'P2X purinoceptor 4' and Ligand = 'BDBM393615'
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM393615(US09969700, 173)
Affinity DataIC50:  54nMAssay Description:Antagonist activity at human P2X4 receptor expressed in HEK cells assessed as reduction in ATP induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM393615(US09969700, 173)
Affinity DataIC50:  64nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influx incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM393615(US09969700, 173)
Affinity DataIC50:  64nMAssay Description:The P2X4 receptor antagonist activity of the compounds of the present invention was measured as follows. The 1321N1 cells stably expressing human P2X...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent