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Found 2 Enz. Inhib. hit(s) with Target = 'P2X purinoceptor 7' and Ligand = 'BDBM50237727'
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50237727(CHEMBL4060938)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at P2X7 receptor in human THP1 cells assessed as inhibition of BzATP-induced YO-PRO-1 Iodide uptake measured every 30 secs for 1 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50237727(CHEMBL4060938)
Affinity DataIC50:  100nMAssay Description:Inhibition of [3H]-Ro- 15-1788 binding to recombinant human gamma-aminobutyric-acid A receptor alpha-2-beta-3-gamma-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed