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Found 2 Enz. Inhib. hit(s) with Target = 'P2Y purinoceptor 1' and Ligand = 'BDBM59704'
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM59704(1-(3,4-dichlorophenyl)-3-[4-[(3,4-dimethyl-1,2-oxa...)
Affinity DataKi:  1.30E+4nMAssay Description:Displacement of [125I]MRS2500 from human P2Y1R expressed in Sf9 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM59704(1-(3,4-dichlorophenyl)-3-[4-[(3,4-dimethyl-1,2-oxa...)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at human P2Y1R expressed in human 1321N1 cells assessed as inhibition of 2-MeSADP-induced increase in intracellular inositol phos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed