Affinity DataKi: 34nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Displacement of [33P]ADP from human recombinant P2Y12 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at human P2Y12 receptor assessed as inhibition of ADP-induced platelet-rich plasma aggregation by turbidimetric methodMore data for this Ligand-Target Pair