TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as inhibition of UDP-induced intracellular calcium mobilization b...More data for this Ligand-Target Pair
TargetP2Y purinoceptor 6(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Compound was tested for inhibition of cathepsin G serine protease to produce one-half maximal enzyme activity.More data for this Ligand-Target Pair
Affinity DataIC50: 2.87E+4nMAssay Description:Histamine H2 receptor antagonistic activity on the isolated spontaneously beating guinea pig right atriumMore data for this Ligand-Target Pair